Major class | Sub-class | Element technology |
---|---|---|
Permeability | Permeability | Caco-2 cells permeability |
MDCK cells permeability | ||
PAMPA membrne Permeability | ||
Plasma protein binding | Plasma protein binding | Plasma protein binding assay |
Drug metabollism | Metabolic stabililty | Plasma stability |
Microsomal stability | ||
Hepatocyte stability | ||
Metabolite profiling & ID | Metabolite profiling & ID | |
Drug metabollism Reaction phenotyping | Reaction phenotyping for CYP (recombinant CYPs) | |
Reaction phenotyping for UGT (recombinant UGTs) | ||
Drug transporter | Drug transporter Reaction phenotyping | Reaction phenotyping for Transport |
Reaction phenotyping for Transport (Kinetic study) | ||
Drug-Drug interaction | Enzyme Inhibition | CYP Inhibition (Screening of CYP inhibition) |
CYP inhibition (IC50 assay) | ||
CYP inhibition (Ki assay) | ||
UGT Inhibition (Screening of UGT inhibition) | ||
UGT Inhibition (IC50 assay) | ||
UGT inhibition (Ki assay) | ||
Time-Dependent Inhibition (IC50 shift assay) | ||
Time-Dependent Inhibition (Kinact/KI assay) | ||
Microsomal binding assay | ||
Transporter Inhibition | Transporter Inhibition (Screening) | |
Transporter Inhibition (IC50 assay) | ||
Transporter Inhibition (Ki assay) | ||
Transporter inhibition (Time-Dependent Inhibition, IC50 shift assay) | ||
Enzyme/Transporter Induction | Enzyme/Transporter Induction | |
Enzyme Induction (EC50 assay) | ||
PXR reporter assay | ||
Cell viability | ||
Bioanalytical services | Bioanalytical service | 약물분석법개발 |
In vivo PK 혈장 분석 | ||
Preclinical study | - | - |
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